| 1 |
KONDO T, MITSUDO TA T A. Metal-catalyzed carbon-sulfur bond formation[J]. Chemical Reviews, 2000, 100(8): 3205-3220.
|
| 2 |
FENG M H,TANG B Q,LIANG S H,et al.Sulfur containing scaffolds in drugs: synthesis and application in medicinal chemistry[J].Current Topics in Medicinal Chemistry, 2016, 16(11): 1200-1216.
doi: 10.2174/1568026615666150915111741
|
| 3 |
ILARDI E A, VITAKU E, NJARDARSON J T. Data-mining for sulfur and fluorine: an evaluation of pharmaceuticals to reveal opportunities for drug design and discovery[J]. Journal of Medicinal Chemistry, 2014, 57(7): 2832-2842.
doi: 10.1021/jm401375q
|
| 4 |
SMITH B R, EASTMAN C M, NJARDARSON J T. Beyond C, H, O, and N! Analysis of the elemental composition of US FDA approved drug architectures[J]. Journal of Medicinal Chemistry, 2014, 57(23): 9764-9773.
doi: 10.1021/jm501105n
|
| 5 |
CINAR M E, OZTURK T. Thienothiophenes, dithienothiophenes, and thienoacenes: syntheses, oligomers, polymers, and properties[J]. Chemical Reviews, 2015, 115(9): 3036-3140.
doi: 10.1021/cr500271a
|
| 6 |
TAKIMIYA K, OSAKA I, MORI T. et al.Organic semiconductors based on Benzothieno[3,2-b]benzothiophene Substructure[J]. Accounts of Chemical Research, 2014, 47:1493-1502.
doi: 10.1021/ar400282g
|
| 7 |
SCOTT K A, NJARDARSON J T. Analysis of US FDA-approved drugs containing sulfur atoms[J]. Topics in Current Chemistry (Cham), 2018, 376(1): 5.
doi: 10.1007/s41061-018-0184-5
|
| 8 |
HAMMOND M L, ZAMBIAS R A, CHANG M N, et al. Antioxidant-based inhibitors of leukotriene biosynthesis. The discovery of 6-[1-[2-(hydroxymethyl)phenyl]-1-propen-3-yl]-2, 3-dihydro-5-benzofuranol, a potent topical antiinflammatory agent[J]. Journal of Medicinal Chemistry, 1990, 33(3): 908-918.
doi: 10.1021/jm00165a005
|
| 9 |
KATRITZKY A R, ZHANG Z X, LAN X F. et al. O-(α-Benzotriazolylalkyl)phenols: Novel precursors for the preparation of ortho-substituted phenols via intermediate o-quinone methides[J]. Journal of Organic Chemistry, 1994, 59(7):1900-1903.
doi: 10.1021/jo00086a050
|
| 10 |
MODICA E, ZANALETTI R, FRECCERO M, et al. Alkylation of amino acids and glutathione in water by o-quinone methide. Reactivity and selectivity[J]. The Journal of Organic Chemistry, 2001, 66(1): 41-52.
|
| 11 |
SHAIKH A K, COBB A J A, VARVOUNIS G. Mild and rapid method for the generation of ortho-(naphtho)quinone methide intermediates[J]. Organic Letters, 2012, 14(2): 584-587.
doi: 10.1021/ol203196n
|
| 12 |
LAU C K, WILLIAMS H W R, TARDIFF S, et al. ortho-Specific alkylation of phenols via 1, 3, 2-benzodioxaborins[J]. Canadian Journal of Chemistry, 1989, 67(9): 1384-1387.
doi: 10.1139/v89-212
|
| 13 |
GUO W G, WU B, ZHOU X. et al. Formal asymmetric catalytic thiolation with a bifunctional catalyst at a water-oil interface: synthesis of benzyl thiols[J]. Angewandte Chemie, International Edition, 2015, 54(15):4522-4526.
doi: 10.1002/anie.201409894
|
| 14 |
LAI Z W, SUN J W. Enantioselective addition of thiols to ortho-quinone methides catalyzed by chiral phosphoric acids[J]. Synlett, 2015, 27(4): 555-558.
doi: 10.1055/s-0035-1560546
|
| 15 |
PATHAK T P, SIGMAN M S.Applications of ortho-quinone methide intermediates in catalysis and asymmetric synthesis[J]. Journal of Organic Chemistry, 2011, 76(22):9210-9215.
doi: 10.1021/jo201789k
|
| 16 |
WILLIS N J, BRAY C D. Ortho-quinone methides in aatural product synthesis[J]. Chemistry-A European Journal, 2012, 18(30): 9160-9173.
doi: 10.1002/chem.201200619
|
| 17 |
CARUANA L, FOCHI M, BERNARDI L. The emergence of quinone methides in asymmetric organocatalysis[J]. Molecules, 2015, 20(7): 11733-11764.
doi: 10.3390/molecules200711733
|
| 18 |
MATTSON A E, SCHEIDTK A.Nucleophilic acylation of o-quinone methides: an umpolung strategy for the synthesis of α-aryl ketones and benzofurans[J]. Journal of the American Chemical Society, 2007, 129(15): 4508-4509.
doi: 10.1021/ja068189n
|
| 19 |
LUAN Y, SCHAUS S E. Enantioselective addition of boronates to o-quinone methides catalyzed by chiral biphenols[J]. Journal of the American Chemical Society, 2012, 134(49): 19965-19968.
doi: 10.1021/ja309076g
|
| 20 |
CHEN M W, CAO L L, YE Z S, et al. A mild method for generation of o-quinone methides under basic conditions. The facile synthesis of trans-2, 3-dihydrobenzofurans[J]. Chemical Communications, 2013, 49(16): 1660.
doi: 10.1039/c3cc37800d
|
| 21 |
BAI W J, DAVID J G, FENG Z G, et al. The domestication of ortho-quinone methides[J]. Accounts of Chemical Research, 2014, 47(12): 3655-3664.
doi: 10.1021/ar500330x
|
| 22 |
VAN DE WATER R W,PETTUS T R R.O-quinone methides:Intermediates underdeveloped and underutilized in organic synthesis[J].Tetrahedron, 2002, 58(27): 5367-5405.
doi: 10.1016/S0040-4020(02)00496-9
|
| 23 |
KULIKOV A, ARUMUGAM S, POPIK V V. Photolabile protection of alcohols, phenols, and carboxylic acids with 3-hydroxy-2-naphthalenemethanol[J]. Journal of Organic Chemistry, 2008, 73(19): 7611-7615.
doi: 10.1021/jo801302m
|
| 24 |
张硕, 于一涛, 李庆刚, 等. Sc(Ⅲ)催化硫醇对邻亚甲基苯醌的亲核加成反应合成邻羟基苄硫醚衍生物[J]. 高等学校化学学报, 2019, 40(4): 725-732.
doi: 10.7503/cjcu20180599
|
